Search results for " Oxazines"

showing 6 items of 6 documents

Differential reactivity of fluorinated homopropargylic amino esters vs gold(I) salts. The role of the nitrogen protecting group

2015

The reaction of several homopropargyl amino esters 4, bearing aromatic substituents and a benzyl group as nitrogen substituents, with gold(I) salts gave rise to fluorinated quinolines 6 in a tandem hydroarylation-isomerization process. On the other hand, homopropargyl amino esters 7 containing a carbamate group underwent the carbonyl addition over the triple bond in the presence of gold(I) salts, rendering fluorinated oxazines 8. The use of chiral sulfoxides allowed us to develop the asymmetric version of this protocol. This two processes complete the differential reactivity showed by these types of susbtrates, depending on the nature of the nitrogen protecting group. (C) 2014 Elsevier B.V.…

chemistry.chemical_classificationCarbamateFluorinated alfa-amino acid derivativesAmino estersmedicine.medical_treatmentOrganic ChemistryFluorinated dihydro-quinolineschemistry.chemical_elementOxazinesGold catalysisTriple bondBiochemistryMedicinal chemistryNitrogenInorganic Chemistrychemistry.chemical_compoundchemistrymedicineBenzyl groupEnvironmental ChemistryFluorinated homopropargyl amino estersPhysical and Theoretical ChemistryProtecting groupFluorinated oxazines
researchProduct

A new multi analytical approach for the identification of synthetic and natural dyes mixtures. The case of orcein-mauveine mixture in a historical dr…

2017

In this paper, the application of a multi-analytical approach for the characterisation of synthetic and natural dyes in a historical textile is presented. The work is focused on a historical dress of a Sicilian noblewoman, dating from about 1865–1870. Firstly, SERS on fibre was performed, in order to individuate the classes of dyes employed. The SERS spectra suggested the presence of two main dyes: mauveine and orcein. In order to confirm these preliminary results, two different extraction protocols were applied. The extracts obtained were analysed by ESI-MS, MALDI-ToF and UHPCL-MS analyses, confirming the SERS results. In particular, the application of the ammonia mild extraction technique…

Historynew ammonia extraction methodComplex Mixtureorcein dyeMALDI-ToF; Mauveine; new ammonia extraction method; orcein dyes; SERS on fibre; Sicilian dress; UHPLC-MS; Clothing; Coloring Agents; Complex Mixtures; Female; History 19th Century; Humans; Oxazines; Sicily; Spectrum Analysis; TextilesMALDI-ToF; Mauveine; new ammonia extraction method; orcein dyes; SERS on fibre; Sicilian dress; UHPLC-MS; Analytical Chemistry; Biochemistry; Plant Science; Organic ChemistryMauveineSicilian dreSERS on fibreOxazineColoring agentsPlant ScienceComplex Mixtures01 natural sciencesBiochemistrylaw.inventionAnalytical ChemistryUHPLC-MSClothingUhplc mschemistry.chemical_compoundlawMauveineOxazinesHumansColoring AgentsColoring AgentOrceinSicilySpectrum AnalysiMALDI-ToF19th CenturyChromatographyPolymer science010405 organic chemistryChemistrySpectrum AnalysisTextilesOrganic Chemistryorcein dyesHistory 19th CenturySettore CHIM/06 - Chimica Organica0104 chemical sciencesSicilian dress010404 medicinal & biomolecular chemistryFemaleSpectrum analysismauveine; orcein dyes; Sicilian dress; new ammonia extraction method; SERS on fibre; MALDI-ToF; UHPLC-MSHuman
researchProduct

Nile Red lifetime reveals microplastic identity

2020

Microplastic pollution is recognized as a worldwide environmental problem. The increasing daily use and release of plastics into the environment have led to the accumulation of fragmented microplastics, with potentially awful consequences for the environment, and animal and human health. The detection and identification of microplastics are of utmost importance, but available methods are still limited. In this work, a new approach is presented for the analysis of microplastics based on hydrophobic fluorescence staining with Nile Red, using spectrally resolved confocal fluorescence microscopy and fluorescence lifetime imaging microscopy (FLIM). Significant differences were observed in the em…

MicroplasticsFluorescence-lifetime imaging microscopyMicroplastics010501 environmental sciencesManagement Monitoring Policy and Law01 natural sciences03 medical and health sciencesHuman healthchemistry.chemical_compoundOxazinesFluorescence microscopeAnimalsHumansEnvironmental ChemistryFluorescence staining030304 developmental biology0105 earth and related environmental sciences0303 health sciencesChemistryPublic Health Environmental and Occupational HealthNile redGeneral MedicineFluorescenceSettore FIS/07 - Fisica Applicata(Beni Culturali Ambientali Biol.e Medicin)microplastics nile red fluorescence lifetime Environmental Monitoring Humans Microplastics Oxazines Plastics Water Pollutants ChemicalAquatic environmentBiological systemPlasticsWater Pollutants ChemicalEnvironmental MonitoringEnvironmental Science: Processes & Impacts
researchProduct

FRET multiphoton spectral imaging microscopy of 7-ketocholesterol and Nile Red in U937 monocytic cells loaded with 7-ketocholesterol.

2004

To show the effect of 7-ketocholesterol (7KC) on cellular lipid content by means of flow cytometry and the interaction of 7KC with Nile Red (NR) via ultraviolet fluorescence resonance energy transfer (FRET) excitation of NR on U937 monocytic cells by means of 2-photon excitation confocal laser scanning microscopy (CLSM).Untreated and 7KC-treated U937 cells were stained with NR and analyzed by flow cytometry and CLSM. 3D sequences of images were obtained by spectral analysis in a 2-photon excitation CLSM and analyzed by the factor analysis of medical image sequences (FAMIS) algorithm, which provides factor curves and images. Factor images are the result of the FAMIS image processing method, …

MESH: Cell DeathMESH: Fluorescence Resonance Energy TransferMESH: Mitochondria[SDV.IB.IMA]Life Sciences [q-bio]/Bioengineering/ImagingMESH : Flow CytometryMESH: Flow CytometryMESH: U937 CellsMESH: MonocytesMonocytesMembrane PotentialsMESH : Staining and LabelingMESH : Microscopy Fluorescence MultiphotonOxazinesFluorescence Resonance Energy TransferImage Processing Computer-AssistedHumansMESH: Membrane PotentialsMESH: Microscopy ConfocalMESH : Membrane PotentialsMESH : Fluorescent DyesMESH : Microscopy ConfocalKetocholesterols[ SDV.IB.IMA ] Life Sciences [q-bio]/Bioengineering/ImagingFluorescent DyesMESH : KetocholesterolsMicroscopy ConfocalMESH: HumansMESH : OxazinesCell DeathStaining and LabelingMESH : HumansMESH: KetocholesterolsU937 CellsFlow CytometryMESH: Fluorescent DyesMESH: Image Processing Computer-AssistedMitochondriaMESH: Staining and Labeling[SDV.IB.IMA] Life Sciences [q-bio]/Bioengineering/ImagingMicroscopy Fluorescence MultiphotonMESH : MonocytesMESH : Fluorescence Resonance Energy TransferMESH : Cell DeathMESH : U937 CellsMESH: Microscopy Fluorescence MultiphotonMESH : MitochondriaMESH: OxazinesMESH : Image Processing Computer-Assisted
researchProduct

Deconvolution procedure of the UV-vis spectra. A powerful tool for the estimation of the binding of a model drug to specific solubilisation loci of b…

2015

UV-vis-spectra evolution of Nile Red loaded into Tween 20 micelles with pH and [Tween 20] have been analysed in a non-conventional manner by exploiting the deconvolution method. The number of buried sub-bands has been found to depend on both pH and bio-surfactant concentration, whose positions have been associated to Nile Red confined in aqueous solution and in the three micellar solubilisation sites. For the first time, by using an extended classical two-pseudo-phases-model, the robust treatment of the spectrophotometric data allows the estimation of Nile Red binding constant to the available loci. Hosting capability towards Nile Red is exalted by the pH enhancement. Comparison between bin…

Atomic and Molecular Physics and OpticOxazineAnalytical chemistrySpecific solubilisation lociTween 20PolysorbatesDeconvolutionNile RedMicelleSpectral lineUV-vis spectraAnalytical ChemistrySurface-Active Agentchemistry.chemical_compoundSurface-Active AgentsUltraviolet visible spectroscopycmc; Deconvolution; Nile Red; Specific solubilisation loci; Tween 20; UV-vis spectra; Binding Sites; Oxazines; Polysorbates; Solubility; Spectrophotometry Ultraviolet; Surface-Active Agents; Micelles; Instrumentation; Atomic and Molecular Physics and Optics; Analytical Chemistry; Spectroscopy; Medicine (all)Pulmonary surfactantOxazinesInstrumentationSpectroscopyMicellesAqueous solutionBinding SitesChemistryMedicine (all)Nile redBinding SiteBinding constantAtomic and Molecular Physics and OpticsPolysorbateSolubilitycmcSpectrophotometry UltravioletDeconvolutionMicelle
researchProduct

Durability of Dolutegravir-Based Regimens: A 5-Year Prospective Observational Study

2021

This study evaluates the frequency and causes of dolutegravir (DTG) discontinuation along 5 years of follow-up, in both antiretroviral treatment (ART)-naive and experienced people living with HIV (PLWH). This is a prospective multi-center cohort study enrolling PLWH on DTG from July 2014 until November 2020. DTG-durability was investigated using the Kaplan-Meier survival curve. The Cox proportional-hazards model was used for estimating the hazard ratio (HR) of DTG discontinuation for any cause, and for adverse events (AEs). Nine hundred sixty-three PLWH were included, 25.3% were women and 28.0% were ART-naive. Discontinuations for any causes were 10.1 [95% confidence interval (95% CI) 8.9-1…

adverse events; dolutegravir; durability; HIV; safety; toxicity; virolgical failure; Cohort Studies; Female; Heterocyclic Compounds 3-Ring; Humans; Middle Aged; Oxazines; Piperazines; Prospective Studies; Pyridones; Anti-HIV Agents; HIV InfectionssafetyPediatricsmedicine.medical_specialtySettore MED/17 - Malattie InfettivePyridonesAnti-HIV AgentsOxazineHuman immunodeficiency virus (HIV)adverse eventHIV Infectionsvirolgical failurePyridonemedicine.disease_cause3-RingHIV Infections.PiperazinesCohort Studieschemistry.chemical_compoundHeterocyclic CompoundsHIV; adverse events; dolutegravir; durability; safety; toxicity; virolgical failureOxazinesAntiretroviral treatmentMedicineHumansProspective StudiesAdverse effectPiperazinebusiness.industryPublic Health Environmental and Occupational HealthHIVtoxicityAnti-HIV AgentMiddle Agedadverse eventsDiscontinuationdolutegravirvirolgical failure.Prospective StudieInfectious DiseaseschemistryDolutegravirdurabilityObservational studyFemaleCohort StudiebusinessHeterocyclic Compounds 3-RingHuman
researchProduct